A copper-catalysed amidation of aldehydes via N-hydroxysuccinimide ester formation.

نویسندگان

  • Monica Pilo
  • Andrea Porcheddu
  • Lidia De Luca
چکیده

A copper-catalysed oxidative amidation of aldehydes via N-hydroxysuccinimide ester formation is reported. The methodology employed to prepare amides directly from aldehydes has a very wide scope, is high yielding, and does not need dry conditions. This cross-coupling reaction appears to be simple and makes use of cheap, abundant and easily available reagents.

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عنوان ژورنال:
  • Organic & biomolecular chemistry

دوره 11 47  شماره 

صفحات  -

تاریخ انتشار 2013